Exemestanex is a new generation of drug that blocks enzymes responsible for aromatisation. Exemestanex is significantly different from drugs belonging to the class of aromatase inhibitors. Exemestanex is a better drug. Familiar aromatase inhibitors have only a temporary efficiency, but Exemestanex has an irreversible and permanent effect. As a result of the drug are suppressed 85% or more estrogens in the body of the athlete.
Exemestanex during steroid cycle prevents the side effects that steroids can cause – flavoring. It should be noted that the effect of Exemestanex is fundamentally different from the usual action of Nolvadex for many athletes. It is known that Tamoxifen has no effect on the aromatization process. It just begins to interact with the cellular estrogen receptors, preventing estrogen to join them and form a bond.
Exemestanex also acts on the process of flavoring and suppresses it. Exemestanex structure is very similar to a naturally occurring steroid – androstenedione. Exemestanex principle of operation is that it irreversibly binds to active enzymes hormones. As a result, hormones lose their activity. Exemestanex has no estrogenic or progestogenic activity. But it is characterized by mild androgenic activity.
Breast cancer in postmenopausal women (natural or induced), progressing against the background of antiestrogen therapy, non-steroidal aromatase inhibitors or progestins.
Dosage for men – 12.5-25 mg/day, dosage for Women – 12.5 mg/day
Exemestanex side effects may occur frequently and in varying degrees. For example, an athlete may face unpleasant consequences such as: nausea, fatigue, sweating, dizziness, headache, skin rash, insomnia, etc.